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4-Amino-7-chloroquinolines: Probing Ligand Efficiency Provides Botulinum Neurotoxin Serotype A Light Chain Inhibitors with Significant Antiprotozoal Activity
(Amer Chemical Soc, Washington, 2013)
Structurally simplified analogues of dual antimalarial and botulinum neurotoxin serotype A light chain (BoNT/A LC) inhibitor bis-aminoquinoline (1) were prepared. New compounds were designed to improve ligand efficiency ...
Investigation of nanocrystalline phases in Li-La-Fe-O system formed by the decomposition of acetylacetonato complexes
(Elsevier Science Sa, Lausanne, 2007)
Applying a new synthesis route based on the thermal decomposition of a mixture acetylacetonato complexes, Li(AA), La(AA)(3) and Fe(AA)(3), Li, La ferrite (Li0.5La0.08Fe2.42O4) was formed. The element analysis performed by ...
Structure, configuration, conformation and quantification of the push pull-effect of 2-alkylidene-4-thiazolidinones and 2-alkylidene-4,5-fused bicyclic thiazolidine derivatives
(Pergamon-Elsevier Science Ltd, Oxford, 2010)
Structures of a series of push-pull 2-alkylidene-4-thiazolidinones and 2-alkylidene-4,5-fused bicyclic thiazolidine derivatives were optimized at the B3LYP/6-31G(d) level of theory in the gas phase and discussed with respect ...
Formal Synthesis of (-)-Oseltamivir Phosphate
(Georg Thieme Verlag Kg, Stuttgart, 2013)
The formal synthesis of (-)-oseltamivir phosphate (Tamiflu (TM)) was accomplished starting from (S)-pyroglutamic acid. The synthesis comprised two carbon-carbon bond forming reactions, the first one being a diastereoselective, ...
Electrospray mass spectrometric studies of a potential antitumor drug and its analogous platinum(II) and platinum(IV) complexes with the ethylenediamine-N,N '-di-3-propanoato ligand and its dibutyl ester
(Springer Wien, Wien, 2009)
The electrospray mass spectrometric (ESI-MS) behavior of the complexes trans-dichloro(ethylenediamine-N, N'-di-3-propionato) platinum(IV), trans-dibromo(ethylenediamine-N, N'-di-3-propionato) platinum( IV), dichloro ...
pH-Dependent Leaching of Dump Coal Ash-Retrospective Environmental Analysis
(Taylor & Francis Inc, Philadelphia, 2009)
Trace and major elements in coal ash particles from dump of "Nikola Tesla A" power plant in Obrenovac near Belgrade (Serbia) can cause pollution, due to leaching by atmospheric and surface waters. In order to assess this ...
Different intermolecular interactions in azido[2-(diphenylphosphino)benzaldehyde semicarbazonato-kappa P-2,N-1,O]nickel(II)
(Wiley-Blackwell, Malden, 2009)
The title compound, [Ni(C20H17N3OP)(N-3)], is the first complex with a semicarbazide-based ligand having a P atom as one of the donors. The influence of the P atom on the deformation of the coordination geometry of the ...
Stabilizing non-covalent interactions of ligand aromatic moieties and proline in ligand-protein systems
(Springer Wien, Wien, 2015)
Proline, due to its conformational specificity, is known to show some unique properties and has significant functions in the tertiary structure of proteins. It was suggested that proline could have an important influence ...
Different effects of pentobarbital and pentylenetetrazol on nitric oxide levels in rat frontal cortex / Uticaj pentobarbitala i pentilenetetrazola na nivo azot oksida u frontalnom korteksu pacova
(De Gruyter Open Ltd, Warsaw, 2005)
Levels of nitric oxide (NO) in the rats frontal cortex were continuously monitored before and after intraperitoneal administration of an antiepileptic drug-pentobarbital (20 and 40 mg/kg) or convulsant drug - pentylenetetrazol ...
Emission of Polycyclic Aromatic Hydrocarbons from Beech Wood Combustion
(Taylor & Francis Inc, Philadelphia, 2013)
This study reports results on 16 EU priority polycyclic aromatic hydrocarbons in smoke produced by beech wood combustion from Zlatibor region, Serbia. Smoke samples were collected with two different types of tubes (PUF and ...